BiochemistrybioRxiv
A distributed residue network permits conformational binding specificity in a conserved family of actin remodelers
T. Hwang, S. S. Parker, S. M. Hill…·A. E. Keating
The paper identifies a conformational mechanism enabling specificity in ENAH EVH1 binding to PCARE, and designs a highly selective inhibitor.
DOI 10.7554/elife.70601