Development of a Triazolobenzodiazepine-Based PET Probe for Subtype-Selective Vasopressin 1A Receptor Imaging
A. Haider, Z. Xiao, X. Xia, J. Chen, R. S. Van, S. Kuang, C. Zhao, J. Rong, T. Shao, P. Ramesh, A. Aravind, Y. Shao, C. Ran, L. Young, S. H. Liang
This paper develops a PET probe for subtype-selective V1A receptor imaging in peripheral organs, showing high affinity and selectivity for V1A over other vasopressin receptors.
bioRxiv · Feb 9, 2021Pharmacology & Toxicology