Cancer BiologybioRxiv
Covalent Disruptor of YAP-TEAD Association Suppresses Defective Hippo Signaling
M. Fan, W. Lu, J. Che…·N. Gray
This paper develops a covalent inhibitor of the YAP-TEAD complex, demonstrating its ability to suppress Hippo signaling defects and inhibit cancer cell growth.
DOI 10.7554/elife.78810