BiochemistrybioRxiv
Targeting the Pregnane X Receptor Using Microbial Metabolite Mimicry
Z. Dvorak, F. Felix Kopp, C. M. Costello…·R. B. Sartor
This paper develops FKK6, a non-cytotoxic PXR agonist derived from microbial metabolite mimicry, which reduces inflammation and validates the strategy for drug discovery.
DOI 10.15252/emmm.201911621