Pharmacology & ToxicologybioRxivPreprint
Discovery of imidazole-based inhibitors of P. falciparum cGMP-dependent protein kinase
R. R. Yadav, M. L. de Souza, M. L. Gonzalez…·D. P. Rotella
The paper identifies imidazole-based inhibitors of PfPKG with good potency and low hERG activity against multiple Plasmodium species.
DOI 10.1101/2021.11.05.467463