BiochemistrybioRxivPreprint
An acetyl-click screening platform identifies a small molecule inhibitor of Histone Acetyltransferase 1 (HAT1) with anti-tumor activity
J. J. Gruber, A. Rangarajan, T. Chou…·A. M. Lipchik
This paper identifies a small molecule inhibitor of HAT1, a histone acetyltransferase, showing anti-tumor activity in vitro and in vivo.
DOI 10.1101/2021.06.25.449993