Cancer BiologybioRxiv
The Dimer-dependent Catalytic Activity of RAF Family Kinases Is Revealed Through Characterizing Their Oncogenic Mutants
J. Yuan, W. H. Ng, P. Y. P. Lam…·J. Hu
This study identifies dimer-dependent catalytic activity in RAF family kinases through analysis of oncogenic mutants, revealing differential inhibitor resistance and MEK phosphorylation mechanisms.
DOI 10.1038/s41388-018-0365-2