BiochemistrybioRxiv
Bariatric surgery reveals a gut-restricted TGR5 agonist that exhibits anti-diabetic effects
S. N. Chaudhari, D. A. Harris, H. Aliakbarian…·A. S. Devlin
This study identifies CA7S, a gut-restricted TGR5 agonist that improves glucose tolerance in insulin-resistant mice by inducing GLP-1 secretion.