Structural flexibility of apolipoprotein E-derived arginine-rich peptides improves their cell penetration capability
Y. Takechi-Haraya, T. Ohgita, A. Usui, K. Nishitsuji, K. Uchimura, Y. Abe, R. Kawano, M. I. Konaklieva, M. Reimund, A. T. Remaley, Y. Sato, K.-i. Izutsu, H. Saito
This study shows that structural flexibility of A2-17 peptide enhances its ability to penetrate cell membranes compared to its constrained variants.
bioRxiv · Aug 16, 2023Biophysics