PROxAb Shuttle: A non-covalent plug-and-play platform for the rapid generation of tumor-targeting antibody-PROTAC conjugates
H. Schneider, S. Jaeger, D. Koenning, N. Rasche, C. Schroeter, D. Elter, A. Evers, M. Lecomte, F. Riccardi Sirtori, D. Schwarz, A. Wegener, I. Hartung, M. Rieker
This paper introduces a platform for creating tumor-targeting antibody-PROTAC conjugates that enhances bioavailability and specificity without modifying PROTACs or antibodies.
bioRxiv · Sep 29, 2023 · PreprintBiochemistry