Development of radiofluorinated MLN-4760 derivatives for PET imaging of the SARS-CoV-2 entry receptor ACE2
J. Wang, D. Beyer, C. Vaccarin, Y. He, M. Tanriver, R. M. Benoit, X. Deupi, L. Mu, J. W. Bode, r. Schibli, C. Mueller
This paper develops and evaluates radiofluorinated derivatives of MLN-4760 for PET imaging of ACE2, finding that [18F]F-MLN-4760 shows superior binding affinity and yield.
bioRxiv · Mar 20, 2024Pharmacology & Toxicology