BiochemistrybioRxiv
Kinases in motion: impact of protein and small molecule interactions on kinase conformations
V. Kugler, S. Schwaighofer, A. Feichtner…·E. Stefan
This study uses KinCon-reporter technology to analyze conformational changes in disease-associated kinases upon drug, regulatory protein, and pathway activation interactions, revealing insights into therapeutic strategies.
DOI 10.7554/elife.94755.3