BiochemistrybioRxiv
Mavacamten stabilizes a folded-back sequestered super-relaxed state of β-cardiac myosin
R. L. Anderson, D. V. Trivedi, S. S. Sarkar…·J. A. Spudich
The paper shows that mavacamten stabilizes a folded-back sequestered super-relaxed state of β-cardiac myosin, linking mutations to cardiomyopathy mechanisms.
DOI 10.1073/pnas.1809540115